What is Rapastinel?
GLYX 13, also known as Rapastinil, is a partial agonist that targets the glycine site of N-methyl-D-aspartate receptor (NMDAR). It has the characteristic of regulating NMDAR function, activating the receptor to produce physiological responses, and preventing the side effects of receptor overactivation. It has long-lasting antidepressant effects and is approved as an adjuvant therapy for the treatment of refractory severe depression. If you need to consult or order high-quality GLYX 13 products, please contact us.
| Product name | GLYX 13 |
| CAS | 117928-94-6 |
| Molecular formula | C18H31N5O6 |
| Molecular weight | 413.47 |
| EINECS Number | NA |
| melting point | NA |
| solubility | NA |
| Storage conditions | Keep in dark place,Inert atmosphere,Store in freezer, under -20°C |
| Appearance | White powder |
| boiling point | 844.2±65.0 °C |
| Density | 1.370±0.06 g/cm3 |
Product Specification
| Item | Specification | Results |
| Appearance | White to brown powder | White powder |
| purity | ≥98% | 99.12% |
| Odor | Characteristic | Conforms |
| Total Heavy metals | ≤10ppm | 2ppm |
| Total microbacterial count | ≤1000cfu/g | 125cfu/g |
| Yeast &Mould | ≤100cfu/g | 56cfu/g |
| Escherichia Coli presence | Negative | Negative |
| Salmonella | Negative | Negative |
| Staphylococcus | Negative | Negative |
| Conclusion：Conform with enterprise specification. | ||
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Where is Rapastinel usually used?
GLYX 13 is mainly used as an N-methyl-D-aspartate receptor (NMDAR) modulator, with partial agonist properties, and has potential applications in the treatment of depression. Its uniqueness lies in its regulatory effect on NMDA receptors, which can activate the receptors to produce the required physiological responses and to some extent prevent the possible side effects of excessive receptor activation, thus achieving precise regulation of neural signal transduction. This regulatory mechanism provides a theoretical basis for the potential application of rapatinib in the treatment of depression.
In addition, it can exist in different forms, including free form and compound salt form, such as Rapastinel Trifluoroacetate. These two forms have important equivalence in terms of biological activity, which means that at the same molar concentration, their regulatory effects on NMDAR are similar. This equivalence ensures that scientists and doctors can make decisions based on the physical properties of the drug, such as solubility and stability, rather than choosing which form to use based on the drug's biological activity.
In summary, it has great potential in treating neurological disorders, especially in the treatment of depression, which has attracted widespread attention. With the deepening of clinical research and continuous technological advancement, it is expected to become one of the important drugs for treating important diseases such as depression.
What are the effects of Rapastinel?
The GLYX 13 effects include the following:
Antidepressant effect: It exerts antidepressant effects by activating the ERK/mTOR/BDNF/VGF signaling pathway. In phase II clinical and preclinical rodent model studies, it has been found to rapidly and consistently improve depressive symptoms.
Regulating NMDAR function: It can exhibit more subtle and complex patterns of action when regulating NMDAR function, activating receptors to produce the required physiological responses while also preventing potential side effects of receptor overactivation to some extent, providing new possibilities for the treatment of various neurological diseases.
Equivalence of drug forms: It can exist in different forms, which helps to improve the bioavailability of drugs.
In summary, GLYX 13 has shown significant effects in antidepressant treatment and regulation of NMDAR function, and its equivalence in different forms provides flexibility for the preparation of drug formulations.
How and where to buy Rapastinel wholesale?
Our products undergo experimental testing and are recognized by customers.
You can trust our order because we have a good record of selling legal educational drugs.
A variety of shipping methods for you to choose
|
Transportation Time |
Shipping method |
Cargo weight requirements |
Advantage |
|
3-7 days |
DHL, Germany DHL, Germany DPD, |
Suitable for under 50kg. |
We have warehouses in Germany and California, USA, |
|
7-15 days |
By Air |
Suitable for more than 50kg. |
|
|
15-60 days |
By Sea |
Suitable for more than 500kg. |
Send your Inquiry for more details,Click email:sales2@faithfulbio.com or Whatsapp:+86 17782785148 Now.
FAQ：
Q1:How can I contact your company?
A1: You can reach us through the following means:Phone; Email; Visit our Contact Us page on our website for more options.
Q2:Can I purchase this products directly from your company?
A2:Yes, we welcome both B2B (Business-to-Business) and B2C (Business-to-Consumer) customers. Please visit our website or contact us directly for inquiries about product availability and pricing.
Q3:Does your company offer custom synthesis services?
A3:Yes, we provide custom synthesis services for pharmaceutical intermediates and APIs. Contact us with your specific requirements, and our team will be happy to assist you.
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Note: This compound is only used for laboratory research purposes. The US authorities have not evaluated these claims. Before use, please consult your doctor and learn about available research. This product is not intended for the diagnosis, treatment, cure, or prevention of any disease.
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