Product description
Apalutamide powder belongs to the second generation of highly selective androgen receptor antagonists, and its affinity with androgen receptor is more than 5 times that of the first generation androgen receptor antagonists.
Similar to enzalutamide and apalutamide, darolutamide also inhibits androgen receptor translocation to the nucleus. However, darolutamide has much higher binding to the androgen receptor, which leads to stronger suppression of androgen-induced cell growth and androgen receptor mutations.
If you decide to treat prostate cancer with apalutamide and it doesn't work, you may not be able to use other hormone therapies such as abiraterone, Enzalutamide, or Darolutamide. That's because studies have shown that men who have already used one of these drugs don't respond as well to the others.
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COA
| Item | Specification | Results |
| Appearance | White or off-white powder | Off-white powder |
| Identification | By HPLC | Complies |
| Melting Point | 120ºC~130ºC | 126ºC |
| Loss on Drying | ≤1.00% | 0.21% |
| Heavy Metals | ≤ 10ppm | Complies |
| Sulfated Ash | ≤ 0.10% | 0.03% |
| Chlorine Content | 17.5%~19.5% | 19.30% |
| Arsenic Content | ≤ 0.1ppm | 0.09ppm |
| Lead VContent | ≤ 3.0ppm | 0.50ppm |
| Cadmium Content | ≤ 0.1ppm | 0.10ppm |
| Mercury Content | ≤ 0.1ppm | 0.10ppm |
| Microbiological Test | Coliforms:Negative | Negative |
| Salmonella: Negative | Complies | |
| Total plate count: ≤1000 CFU/g | Pass | |
| Yeast&Mold: ≤50 CFU/g | Pass | |
| Related Substances | Impurity A: ≤0.30% | 0.18% |
| Other unknown impurity: ≤0.10% | 0.07% | |
| Total Impurities: ≤0.50% | 0.42% | |
| Assay | ≥ 98.0% | 99.50% |
| Conclusion | Conform with enterprise specification | |
Physical and chemical properties
Density 1.6± 0.1g /cm3
Molecular formula C21H15F4N5O2S
Molecular weight 477.435
Precision mass 477.088257
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Is apalutamide a chemotherapy drug?
It is important to understand that apalutamide is not a traditional chemotherapy drug and has a different way of working. It works by blocking hormones which stops the cancer cells growing and spreading.
What class of drug is apalutamide?
Apalutamide is in a class of medications called androgen receptor inhibitors. It works by blocking the effects of androgen (a male reproductive hormone) to stop the growth and spread of cancer cells.
How good is Apalutamide Powder?
Apalutamide blocks the effect of testosterone on prostate cancer cells. This will usually slow down the growth of cancer cells. This can help control advanced prostate cancer or delay the spread of localised prostate cancer or locally advanced prostate cancer to other parts of the body.
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why choose us
Our Factory
Package
Shipping Methods
|
Transportation Time |
Shipping method |
Cargo weight requirements |
Advantage |
|
3-7 days |
DHL,Germany DHL,Germany DPD, |
Suitable for under 50kg. |
We have warehouses in Germany and California, USA, and customers in Europe and America can enjoy sending goods directly from these two places. |
|
7-15 days |
By Air |
Suitable for more than 50kg. |
|
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15-60 days |
By Sea |
Suitable for more than 500kg. |
Send your Inquiry for more details, Click email：sales4@faithfulbio.com
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