99% Iloperidone Powder CAS 133454-47-4

HP 873 is a derivative of piperidinyl benzothiazole, pure Fanapt is a white to off white crystalline powder that is almost insoluble in water, slightly soluble in hydrochloric acid, and easily soluble in chloroform, ethanol, methanol, and acetonitrile. In vitro and in vivo experiments have shown that 98% ILOPERIDONE Powder has pharmacological properties similar to other atypical antipsychotic drugs, namely selective effects on the midbrain margin and antipsychotic symptoms, resulting in a low incidence of EPS.

What are the pharmacological effects of ILOPERIDONE?

98% ILOPERIDONE powder mainly exerts therapeutic effects on positive and negative symptoms by blocking D2, D3, 5-HT2A, and norepinephrine (NE) alpha 1/alpha 2C receptors. Blocking these receptors also helps improve patients' emotional disorders and cognitive function. Clinical studies have found that HP-873 has good affinity for multiple receptors of serotonin (5-HT), dopamine (DA), and alpha adrenergic receptors, especially for 5-HT2A receptors, which is 10 times higher than for D2 receptors. At present, experimental evidence has shown that the activity of Fanapt in the limbic system is 300 times higher than that in the substantia nigra striatum. This leads to the fact that this product can not only reduce dopamine activity in the limbic system of the brain to alleviate negative symptoms, but also increase dopaminergic activity in the frontal cortex to improve negative symptoms and cognitive impairment. In addition, Hot sales ILOPERIDONE has a lower affinity for histamine H1 receptors, resulting in a lower risk of excessive sedation or increased body weight. Iloperidone raw material has a low affinity for M1 receptors, so it is less likely to cause anticholinergic adverse reactions, including cognitive dysfunction and gastrointestinal disorders.

What are the side effects of this product?

Compared with common products in the current market, both short-term and long-term safety tests have shown that 98% ILOPERIDONE Powder has fewer adverse reactions. Especially, the induction of extrapyramidal symptoms is relatively rare. The clinical research results show that this product has good safety and tolerance, and its metabolism is good. It is mainly discharged through liver metabolism, and will not induce diabetes. The most common adverse reactions are dizziness, dry mouth, fatigue, nasal congestion, orthostatic hypotension, drowsiness, increased heart rate, weight gain, and QT interval prolongation. However, this product is not very friendly to Alzheimer's disease.

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